Targeting of Histidine Residues to Increase the Pool of Potential Targets Amendable for Covalent Drug Discovery
Time: 3:00 pm
day: Conference Day One
Details:
- Showcasing how to identify and map histidine residues across a wide range of proteins to determine their potential as covalent drug targets
- How to marry the right electrophiles with histidine moieties
- Ligand-first versus electrophile-first approaches to target Histidine residues
