Specific Covalent Targeting of Histidine, Tyrosine & Lysine to Expand the Druggable Proteome
Time: 2:30 pm
day: Conference Day One
Details:
- Development of novel warheads for covalent screening of histidine, tyrosine and lysine residues
- Enhancing the capture and mass spectrometry detection of sensitive peptide-ligand pairs
- Integration of structural information to prioritize novel binding pockets for further development of covalent or non-covalent compounds
