Covalent Fragment-Based Ligand Discovery to Drug Refractory Targets

Time: 5:00 pm
day: Conference Day One

Details:

  • How can covalent fragment-based ligand discovery be leveraged to tackle so-called undruggable targets?
  • What are the advantages of a target-centric approach to covalent fragment-based ligand discovery?
  • What approaches (biochemical and cell-based) can be deployed to progress covalent fragment starting points to mature lead molecules within a drug discovery campaign? 

Speakers: