Round Table: Investigating the Feasibility of Targeting Non-Cysteine Residues & Developing Rational Strategies to Drug New Target
Time: 12:30 pm
day: Day One
Details:
- Evaluating the suitably of non-cysteine residues for covalent targeting to assess feasibility of drugging novel proteins
- Exploring the technological advancements required to effectively identify and target alternative amino acids
- Optimizing warhead selectivity and potency to enable precise targeting whilst mitigating against off-target activity
