Complementary Strategies for Covalent Hit Finding & Characterization
Time: 2:30 pm
day: Day One
Details:
- Strategic application of labelling- vs. function-first approaches for covalent hit finding in vitro and in cells
- Chemoproteomics applications for hit characterization and determination of novel ligandable sites on targets of interest
- Library considerations for covalent hit finding at Novartis